- [1]The semi-synthesis, biological evaluation and docking analysis of the oxime, hydrazine and hydrazide derivatives of platensimycin[J].MedChemComm, 2018
- [2]Semisynthesis of platensimycin derivatives with antibiotic activities in mice via Suzuki–Miyaura cross-coupling reactions[J].Journal of medicinal chemistry, 2018
- [3]Late-stage functionalization of platensimycin leading to multiple analogues with improved antibacterial activity in vitro and in vivo[J].Journal of medicinal chemistry, 2019
- [4]Novel bisubstrate inhibitors for protein N-terminal acetyltransferase D[J].Journal of medicinal chemistry, 2021
- [5]Morphing Natural Product Platensimycin via Heck, Sonogashira, and One-Pot Sonogashira/Cycloaddition Reactions to Produce Antibiotics with In Vivo Activity[J].Antibiotics, 2022
- [6]Venglustat inhibits protein N-terminal methyltransferase 1 in a substrate-competitive manner[J].Journal of Medicinal Chemistry, 2022
- [7]Structure–activity relationship studies of Venglustat on NTMT1 inhibition[J].Journal of Medicinal Chemistry, 2023
- [8]Comparative Study of Adenosine Analogs as Inhibitors of Protein Arginine Methyltransferases and a Clostridioides difficile-Specific DNA Adenine Methyltransferase[J].ACS Chemical Biology, 2023
- [9]Venglustat Analogues with Enhanced Inhibition for Protein N-Terminal Methyltransferases 1/2[J].Journal of Pharmacology and Experimental Therapeutics 385 (S3), 2023
- [10]A unique binding pocket induced by a noncanonical SAH mimic to develop potent and selective PRMT inhibitors[J].Acta Pharmaceutica Sinica B, 2023
| |