Journal Publications

• [1]J.-A, Xiao, J. Li, P.-J. Xia, Z.-F. Zhou, Z.-X. Deng, H.-Y. Xiang, X.-Q. Chen and H. YangDiastereoselective Intramolecular 3+2 -Annulation of Donor-Acceptor Cyclopropane with Imine-Assembling Hexahydropyrrolo 3,2-c quinolinone Scaffolds.Journal of Organic Chemistry, 2016, 81 (22) : 11185-11194.
• [2]P.-J, Xia, J.-A. Xiao, Y.-H. Sun, J. Li, H.-Y. Xiang, X.-Q. Chen and H. YangDivergent Aerobic Oxidative Ring-Opening Cascades of Isatins with 1,2,3,4-Tetrahydroisoquinoline.European Journal of Organic Chemistry, 2016, 2016 (30) : 5096-5101.
• [3]Y, Zheng, J. Wang, P.-J. Xia, Q.-l. Zhao, J.-A. Xiao, H.-Y. Xiang, X.-Q. Chen and H. YangOrganocatalytic Asymmetric Allylic Alkylation of Morita-Baylis-Hillman Carbonates with Diethyl 2-Aminomalonate Assisted by In Situ Protection.Journal of Organic Chemistry, 2017, 82 (23) : 12202-12208.
• [4]Q, Zhao, H. Xiang, J.-A. Xiao, P.-J. Xia, J.-J. Wang, X. Chen and H. YangSelectfluor-Triggered Tandem Cyclization of o-Hydroxyarylenaminones To Access Difluorinated 2-Amino-Substituted Chromanones.Journal of Organic Chemistry, 2017, 82 (18) : 9837-9843.
• [5]H, Xiang, Q. Zhao, Z. Tang, J. Xiao, P. Xia, C. Wang, C. Yang, X. Chen and H. YangVisible-Light-Driven, Radical-Triggered Tandem Cyclization of o-Hydroxyaryl Enaminones: Facile Access to 3-CF2 /CF3-Containing Chromones.Organic Letters, 2017, 19 (1) : 146-149.
• [6]S.-S, Wen, Z.-F. Zhou, J.-A. Xiao, J. Li, H. Xiang and H. YangFacile oxidative cyclization to access C2-quaternary 2-hydroxy-indolin-3-ones: synthetic studies towards matemone.New Journal of Chemistry, 2017, 41 (20) : 11503-11506.
• [7]S, Wang, J. Xiao, J. Li, H. Xiang, C. Wang, X. Chen, R. G. Carter and H. YangDiscovery of temperature-dependent, autoinductive reversal of enantioselectivity: palladium-mediated 3+3 -annulation of 4-hydroxycoumarins.Chemical Communications, 2017, 53 (32) : 4441-4444.
• [8]C.-M, Wang, P.-J. Xia, J.-A. Xiao, J. Li, H.-Y. Xiang, X.-Q. Chen and H. YangPhotoredox-Catalyzed Reductive Dimerization of Isatins and Isatin-Derived Ketimines: Diastereoselective Construction of 3,3'-Disubstituted Bisoxindoles.Journal of Organic Chemistry, 2017, 82 (7) : 3895-3900.
• [9]J.-W, Ren, J. Wang, J.-A. Xiao, J. Li, H.-Y. Xiang, X.-Q. Chen and H. YangL-Pyroglutamic Sulphonamide as Hydrogen-Bonding Organocatalyst: Enantioselective Diels-Alder Cyclization to Construct Carbazolespirooxindoles.Journal of Organic Chemistry, 2017, 82 (12) : 6441-6449.
• [10]Y.-L, Qian, P.-J. Xia, J. Li, Q.-L. Zhao, J.-A. Xiao, H.-y. Xiang and H. YangDiversity-driven and facile 1,3-dipolar cycloaddition to access dispirooxindole-imidazolidine scaffolds.Organic & Biomolecular Chemistry, 2017, 15 (41) : 8705-8708.
• [11]F.-L, Liu, C.-Q. Li, H.-Y. Xiang and S. FengA practical and step-economic route to Favipiravir.Chemical Papers, 2017, 71 (11) : 2153-2158.
• [12]J, Li, X. Zhang, H. Xiang, L. Tong, F. Feng, H. Xie, J. Ding and C. YangC-H Trifluoromethylation of 2-Substituted/Unsubstituted Aminonaphthoquinones at Room Temperature with Bench-Stable (CF3SO2)(2)Zn: Synthesis and Antiproliferative Evaluation.Journal of Organic Chemistry, 2017, 82 (13) : 6795-6800.
• [13]J, Li, J.-A. Xiao, S.-J. Zhao, H.-Y. Xiang and H. YangFacile Construction of Pyrrolo 1,2-a indolenine Scaffold via Diastereoselective 3+2 Annulation of Donor-Acceptor Cyclopropane with Indolenine.Synthesis-Stuttgart, 2017, 49 (18) : 4292-4298.
• [14]J, Li, S.-S. Wang, P.-J. Xia, Q.-L. Zhao, J.-A. Xiao, H.-Y. Xiang, X.-Q. Chen and H. YangUnusual Ligand-to-Metal-Ratio-Controlled Bidirectional Enantioselectivity in Pd-Catalysed 3+3 -Annulation of Morita-Baylis-Hillman Acetate.European Journal of Organic Chemistry, 2017, 2017 (46) : 6961-6965.
• [15]Q.-L, Zhao, H.-Y. Xiang, C.-H. Yang, J.-A. Xiao, P.-J. Xia, X.-Q. Chen and H. YangStraightforward Synthesis of Novel Difluorinated 2-Hydroxyl-Substituted Dihydroquinolones Through Selectfluor-triggered Annulation of 2-Aminoarylenaminones.Chemistryselect, 2018, 3 (32) : 9218-9221.
• [16]H, Xiang, Q.-L. Zhao, P.-J. Xia, J.-A. Xiao, Z.-P. Ye, X. Xie, H. Sheng, X.-Q. Chen and H. YangVisible-Light-Induced External Radical-Triggered Annulation To Access CF2-Containing Benzoxepine Derivatives.Organic Letters, 2018, 20 (5) : 1363-1366.
• [17]H, Xiang, X. Wang, Y. Chen, X. Zhang, Y. Chen, C. Tan, Y. Wang, J. Ding, L.-H. Meng and C. YangDiscovery of clinical candidate methyl (5-(6-((4(methylsulfonyl)piperazin-1-yl)methyl)-4-morpholinopyrrolo 2,1- f 1,2,4 triazin-2-yl)-4-(trifluoromethyl)pyridin-2-yl)carbamate (CYH33) : A highly potent and selective PI3K alpha inhibitor for the treatment of advanced solid tumors.Cancer Research, 2018, 78 (13)
• [18]P.-J, Xia, J. Li, Y.-L. Qian, Q.-L. Zhao, H.-Y. Xiang, J.-A. Xiao, X.-Q. Chen and H. YangSolvent-Minimized, Chromatography-Free, Diastereoselective Synthesis of Oxazolidine-Dispirooxindoles via oxa-1,3-Dipolar Cycloaddition of 3-Oxindole.Journal of Organic Chemistry, 2018, 83 (5) : 2948-2953.
• [19]J, Wang, Z.-X. Deng, C.-M. Wang, P.-J. Xia, J.-A. Xiao, H.-Y. Xiang, X.-Q. Chen and H. YangUnraveling and Manipulating the Stereospecific Retro-Aldol Reaction in the Organocatalytic Asymmetric Aldol Reaction of Isatin and Cyclohexanone.Organic Letters, 2018, 20 (23) : 7535-7538.
• [20]C.-M, Wang, D. Song, P.-J. Xia, Z.-P. Ye, J.-A. Xiao, H.-Y. Xiang, X.-Q. Chen and H. YangPhotoredox-catalyzed direct aminoalkylation of isatins: diastereoselective access to 3-hydroxy-3-aminoalkylindolin-2-ones analogues.Organic Chemistry Frontiers, 2018, 5 (10) : 1608-1612.